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9 µM by directly binding to CBP's KIX domain (Kd ~8
The erbB protein family
Coleman PJ
PubMed PMID: 30422008
HCT-116 (colon)
GNE-207 P7-4 9 µM by directly bindingGNE 207 is a potent, selective and orally bioavailable inhibitor of the bromodomain of CBP, with an IC50 of 1 nM, exhibits a selectively index of >2500 fold against BRD4 (1). GNE 207 shows excellent CBP potency, with an EC50 of 18 nM for MYC expression in MV 4 11 cells. Product information CAS Number: 2158266 58 9 Molecular Weight: 510. 59 Formula: C29H30N6O3 Chemical Name: 5 {8 [5 acetyl 1 (oxan 4 yl) 1H,4H,5H,6H,7H pyrazolo[4,3 c]pyridin 3
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